Design and Synthesis of Tricyclic JAK3 Inhibitors with Picomolar Affinities as Novel Molecular Probes

Author:

Gehringer Matthias,Pfaffenrot Ellen,Bauer Silke,Laufer Stefan A.

Publisher

Wiley

Subject

Organic Chemistry,General Pharmacology, Toxicology and Pharmaceutics,Molecular Medicine,Drug Discovery,Biochemistry,Pharmacology

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1. Discovery of C-5 Pyrazole-Substituted Pyrrolopyridine Derivatives as Potent and Selective Inhibitors for Janus Kinase 1;Journal of Medicinal Chemistry;2023-05-10

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3. Pharmacology of inhibitors of Janus kinases – Part 2: Pharmacodynamics;JDDG: Journal der Deutschen Dermatologischen Gesellschaft;2022-11-26

4. Three Heterocyclic Rings Fused (5-6-5);Comprehensive Heterocyclic Chemistry IV;2022

5. Portraying molecular modulation and therapeutic aspects of psoriasis: Retrospection and current status;Journal of Molecular Structure;2021-11

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