Structural and Thermodynamic Characterization of the TYK2 and JAK3 Kinase Domains in Complex with CP-690550 and CMP-6

Author:

Chrencik Jill E.,Patny Akshay,Leung Iris K.,Korniski Brian,Emmons Thomas L.,Hall Troii,Weinberg Robin A.,Gormley Jennifer A.,Williams Jennifer M.,Day Jacqueline E.,Hirsch Jeffrey L.,Kiefer James R.,Leone Joseph W.,Fischer H. David,Sommers Cynthia D.,Huang Horng-Chih,Jacobsen E.J.,Tenbrink Ruth E.,Tomasselli Alfredo G.,Benson Timothy E.

Publisher

Elsevier BV

Subject

Molecular Biology,Structural Biology

Reference48 articles.

1. tyk2, prototype of a novel class of non-receptor tyrosine kinase genes;Firmbach-Kraft;Oncogene,1990

2. Murine JAK3 is preferentially expressed in hematopoietic tissues and lymphocyte precursor cells;Gurniak;Blood,1996

3. Putative tyrosine kinases expressed in K-562 human leukemia cells;Partanen;Proc. Natl Acad. Sci. USA,1990

4. Two novel protein-tyrosine kinases, each with a second phosphotransferase-related catalytic domain, define a new class of protein kinase;Wilks;Mol. Cell. Biol.,1991

5. Therapeutic targeting of Janus kinases;Pesu;Immunol. Rev.,2008

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