Phenylthiazole Antibacterial Agents Targeting Cell Wall Synthesis Exhibit Potent Activity in Vitro and in Vivo against Vancomycin-Resistant Enterococci

Author:

Mohammad Haroon1ORCID,Younis Waleed1,Chen Lu2,Peters Christine E.3,Pogliano Joe3,Pogliano Kit3,Cooper Bruce4,Zhang Jianan5,Mayhoub Abdelrahman67ORCID,Oldfield Eric89,Cushman Mark10,Seleem Mohamed N.111

Affiliation:

1. Department of Comparative Pathobiology, Purdue University College of Veterinary Medicine, West Lafayette, Indiana 47907, United States

2. Department of Biochemistry, University of Illinois at Urbana−Champaign, Urbana, Illinois 61801, United States

3. Division of Biological Sciences, University of California, San Diego, La Jolla, California 92093, United States

4. Bindley Bioscience Center, Purdue University, West Lafayette, Indiana 47907, United States

5. School of Molecular and Cellular Biology, University of Illinois at Urbana−Champaign, Urbana, Illinois 61801, United States

6. Department of Pharmaceutical Organic Chemistry, College of Pharmacy, Al-Azhar University, Cairo, 11884, Egypt

7. Biomedical Sciences, University of Science and Technology, Zewail City of Science and Technology, Giza, Egypt

8. Center for Biophysics and Quantitative Biology, University of Illinois at Urbana−Champaign, Urbana, Illinois 61801, United States

9. Department of Chemistry, University of Illinois at Urbana−Champaign, Urbana, Illinois 61801, United States

10. Department of Medicinal Chemistry and Molecular Pharmacology, Purdue University College of Pharmacy and the Purdue Center for Cancer Research, West Lafayette, Indiana 47907, United States

11. Purdue Institute for Inflammation, Immunology, and Infectious Disease, Purdue University, West Lafayette, Indiana 47907, United States

Funder

National Cancer Institute

Science and Technology Development Fund

National Academy of Sciences

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Reference55 articles.

1. Preventing Healthcare-Associated Infections.CDC at Work;Centers for Disease Control and Prevention:Atlanta, 2016; https://www.cdc.gov/washington/~cdcatWork/pdf/infections.pdf(accessed December 5, 2016).

2. Antimicrobial Resistance Global Report on Surveillance 2014;World Health Organization Press:Geneva, 2014; pp1–232.

3. Antibiotic Resistance Threats in the United States, 2013;Centers for Disease Control and Prevention;Atlanta; 2013; pp1–114.

4. Clinical impact of vancomycin-resistant enterococci

5. Management of multidrug-resistant enterococcal infections

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