Design, Synthesis, and Biological Evaluation of Indole Biphenylcarboxylic Acids as PPARγ Antagonists
Author:
Affiliation:
1. Department of Molecular Therapeutics, The Scripps Research Institute, Scripps Florida, 130 Scripps Way #A2A, Jupiter, Florida 33458, United States
Funder
National Institute of Mental Health
Abrams Charitable Trust
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.5b00218
Reference31 articles.
1. Antidiabetic actions of a non-agonist PPARγ ligand blocking Cdk5-mediated phosphorylation
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