Structure-based discovery of new selective small-molecule sirtuin 5 inhibitors-Reference-Cited by-同舟云学术

Structure-based discovery of new selective small-molecule sirtuin 5 inhibitors

Published:2017-08-18 Issue:1 Volume:91 Page:257-268
ISSN:1747-0277
Container-title:Chemical Biology & Drug Design
language:en
Short-container-title:Chem Biol Drug Des

Author:

Liu Sha¹,Ji Sen¹,Yu Zhu-Jun¹,Wang Hua-Li¹,Cheng Xu¹,Li Wei-Jian¹,Jing Li¹,Yu Yamei¹,Chen Qiang¹^ORCID,Yang Ling-Ling²,Li Guo-Bo¹^ORCID,Wu Yong¹^ORCID

Affiliation:

1. Key Laboratory of Drug Targeting and Drug Delivery System of Ministry of Education; West China School of Pharmacy, and Laboratory of Biotherapy and Cancer Center, West China Hospital; West China Medical School; Sichuan University; Chengdu China

2. College of Food and Bioengineering; Xihua University; Sichuan China

Funder

National Natural Science Foundation of China

Sichuan University

China Postdoctoral Science Foundation

Publisher

Wiley

Subject

Molecular Medicine,Biochemistry,Drug Discovery,Pharmacology,Organic Chemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1111/cbdd.13077/fullpdf

Reference34 articles.

1. The chemical biology of sirtuins

2. The many faces of insulin-like peptide signalling in the brain

3. Lysine Propionylation and Butyrylation Are Novel Post-translational Modifications in Histones

4. Sirt5 Is a NAD-Dependent Protein Lysine Demalonylase and Desuccinylase

5. Lysine Glutarylation Is a Protein Posttranslational Modification Regulated by SIRT5

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