Design, synthesis, biological evaluation and molecular docking study of novel urea-based benzamide derivatives as potent poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors-Reference-Cited by-同舟云学术

Design, synthesis, biological evaluation and molecular docking study of novel urea-based benzamide derivatives as potent poly(ADP-ribose) polymerase-1 (PARP-1) inhibitors

Published:2022-12 Issue: Volume:243 Page:114790
ISSN:0223-5234
Container-title:European Journal of Medicinal Chemistry
language:en
Short-container-title:European Journal of Medicinal Chemistry

Author:

Lu Guoqing,Nie Wenxing,Xin Meixiu,Meng Yingfen,Gu Jiayi,Miao Hui,Cheng Xinyi,Chan Albert S.C.,Zou Yong^ORCID

Publisher

Elsevier BV

Subject

Organic Chemistry,Drug Discovery,Pharmacology,General Medicine

Reference42 articles.

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5. Discovery of pamiparib (BGB-290), a potent and selective poly(ADP-ribose) polymerase (PARP) inhibitor in clinical development;Wang;J. Med. Chem.,2020

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