Synthesis, structure–activity relationship and biological evaluation of novel arylpiperzines as α1A/1D-AR subselective antagonists for BPH-Reference-Cited by-同舟云学术

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Synthesis, structure–activity relationship and biological evaluation of novel arylpiperzines as α1A/1D-AR subselective antagonists for BPH

Published:2015-12 Issue:24 Volume:23 Page:7735-7742
ISSN:0968-0896
Container-title:Bioorganic & Medicinal Chemistry
language:en
Short-container-title:Bioorganic & Medicinal Chemistry

Author:

Xu Fang,Chen Hong,Xu Jingyi,Liang Xue,He Xuelan,Shao Binhao,Sun Xianqiang,Li Bing,Deng Xiaoliang,Yuan Mu

Funder

National Science Foundation of Guangdong Province

Science Foundation of Zhejiang Province

Publisher

Elsevier BV

Subject

Organic Chemistry,Clinical Biochemistry,Drug Discovery,Pharmaceutical Science,Molecular Biology,Molecular Medicine,Biochemistry

Reference26 articles.

1. RBx 6198: A novel α1-adrenoceptor antagonist for the treatment of benign prostatic hyperplasia

2. Structure–activity relationships in 1,4-benzodioxan-related compounds. 10. Novel α1-adrenoreceptor antagonists related to openphendioxan: Synthesis, biological evaluation, and α1d computational study

3. Tamsulosin Potently and Selectively Antagonizes Human Recombinant .ALPHA.1A/1D-Adrenoceptors: Slow Dissociation from the .ALPHA.1A-Adrenoceptor May Account for Selectivity for .ALPHA.1A-Adrenoceptor over .ALPHA.1B-Adrenoceptor Subtype

4. The efficacy and safety of terazosin for the treatment of symptomatic BPH

5. 29-Week Doxazosin Treatment in Patients with Symptomatic Benign Prostatic Hyperplasia

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