Tamsulosin Potently and Selectively Antagonizes Human Recombinant .ALPHA.1A/1D-Adrenoceptors: Slow Dissociation from the .ALPHA.1A-Adrenoceptor May Account for Selectivity for .ALPHA.1A-Adrenoceptor over .ALPHA.1B-Adrenoceptor Subtype-Reference-Cited by-同舟云学术

Tamsulosin Potently and Selectively Antagonizes Human Recombinant .ALPHA.1A/1D-Adrenoceptors: Slow Dissociation from the .ALPHA.1A-Adrenoceptor May Account for Selectivity for .ALPHA.1A-Adrenoceptor over .ALPHA.1B-Adrenoceptor Subtype

Published:2012 Issue:1 Volume:35 Page:72-77
ISSN:0918-6158
Container-title:Biological and Pharmaceutical Bulletin
language:en
Short-container-title:Biol. Pharm. Bull.

Author:

Sato Shuichi¹,Hatanaka Toshiki¹,Yuyama Hironori²,Ukai Masashi¹,Noguchi Yukiko¹,Ohtake Akiyoshi¹,Taguchi Katsunari²,Sasamata Masao¹,Miyata Keiji¹

Affiliation:

1. Applied Pharmacology Research Laboratories, Drug Discovery Research, Astellas Pharma Inc.

2. Pharmacology Research Laboratories, Drug Discovery Research, Astellas Pharma Inc.

Publisher

Pharmaceutical Society of Japan

Subject

Pharmaceutical Science,Pharmacology,General Medicine

Link

http://www.jstage.jst.go.jp/article/bpb/35/1/35_1_72/_pdf

Reference28 articles.

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2. 2) Lepor H. Role of alpha-adrenergic blockers in the treatment of benign prostatic hyperplasia. Prostate Suppl., 3(S3), 75—84 (1990).

3. 3) Auffenberg GB, Helfand BT, McVary KT. Established medical therapy for benign prostatic hyperplasia. Urol. Clin. North Am., 36, 443—459, v—vi (2009).

4. 5) Price DT, Schwinn DA, Lomasney JW, Allen LF, Caron MG, Lefkowitz RJ. Identification, quantification, and localization of mRNA for three distinct α₁-adrenergic receptor subtypes in human prostate. J. Urol., 150, 546—551 (1993).

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