Development and Implementation of a High-Throughput High-Content Screening Assay to Identify Inhibitors of Androgen Receptor Nuclear Localization in Castration-Resistant Prostate Cancer Cells

Author:

Johnston Paul A.12,Nguyen Minh M.3,Dar Javid A.34,Ai Junkui3,Wang Yujuan3,Masoodi Khalid Z.35,Shun Tongying6,Shinde Sunita6,Camarco Daniel P.1,Hua Yun1,Huryn Donna M.17,Wilson Gabriela Mustata8,Lazo John S.9,Nelson Joel B.23,Wipf Peter12710,Wang Zhou2311

Affiliation:

1. Department of Pharmaceutical Sciences, School of Pharmacy, University of Pittsburgh, Pittsburgh, Pennsylvania.

2. University of Pittsburgh Cancer Institute, Pittsburgh, Pennsylvania.

3. Department of Urology, School of Medicine, University of Pittsburgh, Pittsburgh, Pennsylvania.

4. Central Laboratory, College of Science, King Saud University, Riyadh, Saudi Arabia.

5. Transcriptomics and Proteomics Lab, Centre for Plant Biotechnology, Sher-e-Kashmir University of Agricultural Sciences and Technology of Kashmir (SKUAST-K), Shalimar, Srinagar, India.

6. Pittsburgh Specialized Application Center, University of Pittsburgh Drug Discovery Institute, Pittsburgh, Pennsylvania.

7. University of Pittsburgh Chemical Diversity Center, Pittsburgh, Pennsylvania.

8. Department of Health Services and Health Administration, College of Nursing and Health Professions, University of Southern Indiana, Evansville, Indiana.

9. Departments of Pharmacology and Chemistry, University of Virginia, Charlottesville, Virginia.

10. Department of Chemistry, University of Pittsburgh, Pittsburgh, Pennsylvania.

11. Department of Pharmacology and Chemical Biology, University of Pittsburgh, Pittsburgh, Pennsylvania.

Publisher

Mary Ann Liebert Inc

Subject

Drug Discovery,Molecular Medicine

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