Molecular modelling design, synthesis and cytotoxic evaluation of certain substituted 2-(3,4,5-triacetoxybenzoylamino)benzo[d]thiazole and 2-(galloylamino)benzo[d]thiazole derivatives having potential topoisomerase-I inhibitory activity-Reference-Cited by-同舟云学术

Molecular modelling design, synthesis and cytotoxic evaluation of certain substituted 2-(3,4,5-triacetoxybenzoylamino)benzo[d]thiazole and 2-(galloylamino)benzo[d]thiazole derivatives having potential topoisomerase-I inhibitory activity

Published:2012-09-07 Issue:6 Volume:28 Page:1331-1345
ISSN:1475-6366
Container-title:Journal of Enzyme Inhibition and Medicinal Chemistry
language:en
Short-container-title:Journal of Enzyme Inhibition and Medicinal Chemistry

Author:

Ismail Mohamed A. H.¹²,Tratrat Christophe³,Haroun Michelyne G.³

Affiliation:

1. Pharmaceutical Chemistry Department, Faculty of Pharmacy, Ain Shams University, Abbassia, Cairo, Egypt

2. Department of Pharmaceutical Chemistry and Quality Control, Faculty of Pharmacy, Kalamoon University, Deir Atia, Damascus, Syria

3. Department of Pharmaceutical Chemistry, Faculty of Pharmacy, Umm Al-Qura University, Mecca, KSA

Publisher

Informa UK Limited

Subject

Drug Discovery,Pharmacology,General Medicine

Link

https://www.tandfonline.com/doi/pdf/10.3109/14756366.2012.716835

Reference33 articles.

1. DNA TOPOISOMERASE POISONS AS ANTITUMOR DRUGS

2. A Novel Pyrrolidinyl PNA Showing High Sequence Specificity and Preferential Binding to DNA over RNA

3. Synthesis of 4( S )-( N -Boc-amino)-2( S / R )-(thymin-1-ylmethyl)-pyrrolidine- N -1-acetic acid: a novel cyclic PNA with constrained flexibility

4. Synthesis and DNA Binding Property of a Novel Peptide Nucleic Acid that Containscis-4-Adeninyl-L-prolinol Unit

5. Poly(ADP-ribosylation) of DNA topoisomerase I from calf thymus.

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