Transition-metal-free direct C-3 cyanation of quinoxalin-2(1H)-ones with ammonium thiocyanate as the “CN” source-Reference-Cited by-全球学者库

Transition-metal-free direct C-3 cyanation of quinoxalin-2(1H)-ones with ammonium thiocyanate as the “CN” source

Published:2020 Issue:1 Volume:7 Page:113-118
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

Wang Jiayang¹²³⁴,Sun Bin¹²³⁴,Zhang Liang⁵²³⁴,Xu Tengwei⁵²³⁴,Xie Yuanyuan⁵²³⁴,Jin Can⁵²³⁴^ORCID

Affiliation:

1. Collaborative Innovation Center of Yangtze River Delta Region Green Pharmaceuticals

2. Zhejiang University of Technology

3. Hangzhou 310014

4. P. R. China

5. College of Pharmaceutical Sciences

Abstract

A practical protocol for TBHP-mediated oxidative C–H cyanation of quinoxalin-2(1H)-ones utilizing ammonium thiocyanate as the cyanide source has been developed under metal free conditions.

Funder

National Natural Science Foundation of China

Zhejiang University of Technology

Publisher

Royal Society of Chemistry (RSC)

Subject

Organic Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2020/QO/C9QO01055F

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5. Antagonism of the GABA Receptor of Dieldrin-Resistant Houseflies by Fipronil and Its Analogues

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