A diversity-oriented synthesis of bioactive benzanilides via a regioselective C(sp2)–H hydroxylation strategy-Reference-Cited by-同舟云学术

A diversity-oriented synthesis of bioactive benzanilides via a regioselective C(sp2)–H hydroxylation strategy

Published:2016 Issue:3 Volume:7 Page:2229-2238
ISSN:2041-6520
Container-title:Chemical Science
language:en
Short-container-title:Chem. Sci.

Author:

Sun Yong-Hui¹²³⁴⁵^ORCID,Sun Tian-Yu⁶⁷⁸⁹¹⁰,Wu Yun-Dong⁶⁷⁸⁹¹⁰,Zhang Xinhao⁶⁷⁸⁹¹⁰^ORCID,Rao Yu¹²³⁴⁵

Affiliation:

1. MOE Key Laboratory of Protein Sciences

2. Department of Pharmacology and Pharmaceutical Sciences

3. School of Medicine and School of Life Sciences

4. Tsinghua University

5. Beijing 100084

6. Lab of Computational Chemistry and Drug Design

7. Key Laboratory of Chemical Genomics

8. Peking University Shenzhen Graduate School

9. Shenzhen 518055

10. China

Abstract

A diversity-oriented synthesis of bioactive benzanilidesviaC(sp²)–H hydroxylation has been studied. The reaction demonstrates excellent regioselectivity, good tolerance of functional groups, and high yields.

Funder

National Natural Science Foundation of China

Ministry of Science and Technology

Publisher

Royal Society of Chemistry (RSC)

Subject

General Chemistry

Link

http://pubs.rsc.org/en/content/articlepdf/2016/SC/C5SC03905C

Reference91 articles.

1. Antimycobacterial Assessment of Salicylanilide Benzoates including Multidrug-Resistant Tuberculosis Strains

2. Structure-activity and cross-resistance evaluations of a series of human immunodeficiency virus type-1-specific compounds related to oxathiin carboxanilide

Cited by 76 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Recent advances in ruthenium‐catalysed aromatic C−H bond oxygenation, nitrogenation and halogenation;ChemistrySelect;2024-02-13

2. CuBr₂-mediated dehydrogenative [4+2] annulation of 1-naphthyl-1,3-indandiones and alkenes;Chemical Communications;2024

3. Iodine-catalyzed intermolecular 1,2-thio (seleno)amination of alkenes with 1,2,3-triazoles and disulfides (diselenides) in air;Organic Chemistry Frontiers;2024

4. Supported Pd-catalyzed ring opening and chemoselective aminocarbonylative coupling of benzoxazoles with aryl iodides;Catalysis Science & Technology;2024

5. Regioselective synthesis of 2-aminophenols from N-arylhydroxylamines;Organic & Biomolecular Chemistry;2024