Multistage rocket: integrational design of a prodrug-based siRNA delivery system with sequential release for enhanced antitumor efficacy

Author:

Jiang Qian12345,Chen Xiaobing1234,Liang Hong1234,Nie Yu1234ORCID,Jin Rongrong1234,Barz Matthias6789,Yue Dong1234,Gu Zhongwei1011124ORCID

Affiliation:

1. National Engineering Research Center for Biomaterials

2. Sichuan University

3. Chengdu

4. P. R. China

5. Department of Pharmacy

6. Institute of Organic Chemistry

7. Johannes Gutenberg-University Mainz Duesbergweg 10-14

8. 55099 Mainz

9. Germany

10. College of Materials Science and Engineering

11. Nanjing Tech University

12. Nanjing 211816

Abstract

The sequential release of siRNA and anticancer drug was realized in a novel dendritic peptide–prodrug.

Funder

National Natural Science Foundation of China

Sichuan University

Publisher

Royal Society of Chemistry (RSC)

Subject

General Engineering,General Materials Science,General Chemistry,Atomic and Molecular Physics, and Optics,Bioengineering

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