Affiliation:
1. Department of Chemistry, FRQNT Centre for Green Chemistry and Catalysis, McGill University, 801 Sherbrooke St. W., Montreal, Quebec H3A 0B8, Canada
Abstract
This review summarizes the most recent advances of metal-free late-stage functionalization (LSF) of pharmaceutically relevant molecules. Particular emphasis is placed on C–H activation as well as the use of endogenous functional groups.
Funder
Canada Research Chairs
Natural Sciences and Engineering Research Council of Canada
Canada Foundation for Innovation
Fonds Québécois de la Recherche sur la Nature et les Technologies
Consejo Nacional de Ciencia y Tecnología
Publisher
Royal Society of Chemistry (RSC)
Cited by
93 articles.
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