Photoactive platinum(iv) complex conjugated to a cancer-cell-targeting cyclic peptide

Author:

Shi Huayun1234ORCID,Wang Qian56789ORCID,Venkatesh V.1234ORCID,Feng Guokai56789ORCID,Young Lawrence S.10234ORCID,Romero-Canelón Isolda123411ORCID,Zeng Musheng56789ORCID,Sadler Peter J.1234ORCID

Affiliation:

1. Department of Chemistry

2. University of Warwick

3. Coventry CV4 7AL

4. UK

5. State Key Laboratory of Oncology in South China

6. Collaborative Innovation Center for Cancer Medicine

7. Sun Yat-Sen University Cancer Center

8. Guangzhou 510060

9. China

10. Medical School

11. School of Pharmacy

Abstract

Conjugate of a cancer-cell targeting cyclic peptide with a photoactive platinum(iv) complex exhibits enhanced photocytotoxicity and cell accumulation.

Funder

Engineering and Physical Sciences Research Council

H2020 European Research Council

University of Warwick

Office of the Royal Society

Publisher

Royal Society of Chemistry (RSC)

Subject

Inorganic Chemistry

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