Enantioselective [3 + 2] annulation of tryptanthrin-derived ketimines and 2-naphthols: access to polycyclic indolo[2,1-<i>b</i>]quinazoline derivatives-Reference-Cited by-同舟云学术

Enantioselective [3 + 2] annulation of tryptanthrin-derived ketimines and 2-naphthols: access to polycyclic indolo[2,1-b]quinazoline derivatives

Published:2024 Issue:7 Volume:11 Page:2002-2007
ISSN:2052-4129
Container-title:Organic Chemistry Frontiers
language:en
Short-container-title:Org. Chem. Front.

Author:

You Yong¹^ORCID,Gan Guo-Ying¹,Li Qun²³,Liu Xiong-Li⁴^ORCID,Zhang Yan-Ping¹,Wang Zhen-Hua¹^ORCID,Zhao Jian-Qiang¹^ORCID,Yuan Wei-Cheng¹^ORCID

Affiliation:

1. Institute for Advanced Study, Chengdu University, Chengdu 610106, China

2. School of Materials and Environmental Engineering, Chengdu Technological University, Chengdu 611730, China

3. College of Materials and Chemistry & Chemical Engineering, Chengdu University of Technology, Chengdu 610059, China

4. Guizhou Engineering Center for Innovative Traditional Chinese Medicine and Ethnic Medicine, College of Pharmacy, Guizhou University, Guiyang 550025, China

Abstract

An efficient method has been disclosed for the highly enantioselective synthesis of optically pure heptacyclic dihydronaphthofuran-fused indolo[2,1-b]quinazoline derivatives.

Funder

National Natural Science Foundation of China

Natural Science Foundation of Sichuan Province

Chengdu University

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/QO/D3QO02125D

Reference41 articles.

1. Isolation of Antifungal Principle Tryptanthrin, from Strobilanthes Cusia O. Kuntze

2. Recent synthetic and medicinal perspectives of tryptanthrin

3. Discovery of Tryptanthrin Derivatives as Potent Inhibitors of Indoleamine 2,3-Dioxygenase with Therapeutic Activity in Lewis Lung Cancer (LLC) Tumor-Bearing Mice

4. An efficient catalyst-free Mukaiyama-aldol reaction of fluorinated enol silyl ethers with tryptanthrin

5. One-pot, four-component synthesis of spiroindoloquinazoline derivatives as phospholipase inhibitors