Directed regioselective arylation of imidazo[1,2-<i>a</i>]pyridine-3-carboxamides using Rh(<scp>iii</scp>) catalysis-Reference-Cited by-同舟云学术

Directed regioselective arylation of imidazo[1,2-a]pyridine-3-carboxamides using Rh(iii) catalysis

Published:2024 Issue:35 Volume:22 Page:7121-7127
ISSN:1477-0520
Container-title:Organic & Biomolecular Chemistry
language:en
Short-container-title:Org. Biomol. Chem.

Author:

Jahan Kousar¹²,Sood Mehak¹,Jain Osheen¹^ORCID,Sahoo Subash C.³^ORCID,Bharatam Prasad V.¹^ORCID

Affiliation:

1. Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Sector 67, S. A. S. Nagar, Punjab, India

2. Lloyd Institute of Management and Technology, Plot No.-3, Knowledge Park-II, Greater Noida, Uttar Pradesh, India-201306

3. Department of Chemistry & Centre of Advanced Studies in Chemistry, Panjab University, Chandigarh – 160014, India

Abstract

We introduced, for the first time, N-methoxyamide directed proximal C–H bond activation of imidazo[1,2-a]pyridines for C(sp2)–C(sp2) bond formation via a transition metal catalysed approach to obtain C-5 arylated imidazo[1,2-a]pyridines.

Funder

Department of Biotechnology, Ministry of Science and Technology

Publisher

Royal Society of Chemistry (RSC)

Link

http://pubs.rsc.org/en/content/articlepdf/2024/OB/D4OB01166J

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