Comprehensive assay of kinase catalytic activity reveals features of kinase inhibitor selectivity
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Publisher
Springer Science and Business Media LLC
Link
http://www.nature.com/articles/nbt.2017.pdf
Reference36 articles.
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4. Bain, J. et al. The selectivity of protein kinase inhibitors: a further update. Biochem. J. 408, 297–315 (2007).
5. Davies, S.P., Reddy, H., Caivano, M. & Cohen, P. Specificity and mechanism of action of some commonly used protein kinase inhibitors. Biochem. J. 351, 95–105 (2000).
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