A road map to evaluate the proteome-wide selectivity of covalent kinase inhibitors-Reference-Cited by-同舟云学术

A road map to evaluate the proteome-wide selectivity of covalent kinase inhibitors

Published:2014-07-13 Issue:9 Volume:10 Page:760-767
ISSN:1552-4450
Container-title:Nature Chemical Biology
language:en
Short-container-title:Nat Chem Biol

Author:

Lanning Bryan R,Whitby Landon R,Dix Melissa M,Douhan John,Gilbert Adam M,Hett Erik C,Johnson Theodore O,Joslyn Chris,Kath John C,Niessen Sherry,Roberts Lee R,Schnute Mark E,Wang Chu,Hulce Jonathan J,Wei Baoxian,Whiteley Laurence O,Hayward Matthew M,Cravatt Benjamin F

Publisher

Springer Science and Business Media LLC

Subject

Cell Biology,Molecular Biology

Link

http://www.nature.com/articles/nchembio.1582.pdf

Reference54 articles.

1. Manning, G., Whyte, D.B., Martinez, R., Hunter, T. & Sudarsanam, S. The protein kinase complement of the human genome. Science 298, 1912–1934 (2002).

2. Knight, Z.A. & Shokat, K.M. Features of selective kinase inhibitors. Chem. Biol. 12, 621–637 (2005).

3. Liu, Q. et al. Developing irreversible inhibitors of the protein kinase cysteinome. Chem. Biol. 20, 146–159 (2013).

4. Rosenblum, J.S., Nomanbhoy, T.K. & Kozarich, J.W. Functional interrogation of kinases and other nucleotide-binding proteins. FEBS Lett. 587, 1870–1877 (2013).

5. Krishnamurty, R. & Maly, D.J. Chemical genomic and proteomic methods for determining kinase inhibitor selectivity. Comb. Chem. High Throughput Screen. 10, 652–666 (2007).

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