Identification of amino acid residues responsible for the α5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABAA receptor-Reference-Cited by-同舟云学术

Identification of amino acid residues responsible for the α5 subunit binding selectivity of L-655,708, a benzodiazepine binding site ligand at the GABAA receptor

Published:2001-12-20 Issue:2 Volume:77 Page:445-451
ISSN:0022-3042
Container-title:Journal of Neurochemistry
language:en
Short-container-title:

Author:

Casula M. Anna,Bromidge Frances A.,Pillai Gopalan V.,Wingrove Peter B.,Martin Karine,Maubach Karen,Seabrook Guy R.,Whiting Paul J.,Hadingham Karen L.

Publisher

Wiley

Subject

Cellular and Molecular Neuroscience,Biochemistry

Link

http://onlinelibrary.wiley.com/wol1/doi/10.1046/j.1471-4159.2001.00289.x/fullpdf

Reference23 articles.

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2. International union of pharmacology. XV. Subtypes of gamma-aminobutyric acid (A) receptors: classification on the basis of subunit structure and receptor function;Barnard;Pharmacol. Rev.,1998

3. Residues at positions 206 and 209 of the α1 subunit of γ-aminobutyric acidA receptors influence affinities for benzodiazepine binding site ligands;Buhr;Mol. Pharmacol.,1997

4. Structural requirements for ligand interactions at the benzodiazepine recognition site of the GABA(A) receptor;Davies;J. Neurochem.,1998

5. Cloning of cDNA sequences encoding human α2 and α3 γ-aminobutyric acidA receptor subunits and characterization of the benzodiazepine pharmacology of recombinant α1-, α2-, α3-, and α5-containing human γ-aminobutyric acidA receptors;Hadingham;Mol. Pharmacol.,1993a

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