Highly Potent and Isoform Selective Dual Site Binding Tankyrase/Wnt Signaling Inhibitors That Increase Cellular Glucose Uptake and Have Antiproliferative Activity

Author:

Nathubhai Amit1ORCID,Haikarainen Teemu2,Koivunen Jarkko2,Murthy Sudarshan2,Koumanov Françoise3,Lloyd Matthew D.1,Holman Geoffrey D.3,Pihlajaniemi Taina2,Tosh David3,Lehtiö Lari2,Threadgill Michael D.1

Affiliation:

1. Drug and Target Discovery, Department of Pharmacy and Pharmacology, University of Bath, Claverton Down, Bath, Somerset BA2 7AY, U. K.

2. Faculty of Biochemistry and Molecular Medicine, Biocenter Oulu, University of Oulu, PO Box 5400, 90014 Oulu, Finland

3. Department of Biology and Biochemistry, University of Bath, Bath BA2 7AY, U. K.

Funder

Medical Research Council

Worldwide Cancer Research

Suomen Akatemia

European Synchrotron Radiation Facility

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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