Discovery of Potent and Orally Bioavailable Platelet-Derived Growth Factor Receptor (PDGFR) Inhibitors for the Treatment of Osteosarcoma

Author:

Chen Xiaojing1,Liu Lu1,Liu Peng1,Chen Yingying1,Lin Dan2,Yan Hao1,Yan Qi1,Wang Yi1,Qiu Yinda1,Fang Bo1ORCID,Huang Huijing1,Qian Jianchang1,Zhao Yunjie1,Du Zhou3,Zhang Qianwen1,Li Xiaokun1,Zheng Xiaohui1,Liu Zhiguo1ORCID

Affiliation:

1. Chemical Biology Research Center at School of Pharmaceutical Sciences, Wenzhou Medical University, 1210 University Town, Wenzhou, Zhejiang 325035, People’s Republic of China

2. The Eye Hospital, School of Ophthalmology and Optometry, Wenzhou Medical University, Wenzhou, Zhejiang 325035, People’s Republic of China

3. Department of General Surgery, The First Affiliated Hospital of Wenzhou Medical University, Wenzhou, Zhejiang 325035, People’s Republic of China

Funder

Wenzhou Medical University

National Natural Science Foundation of China

Natural Science Foundation of Zhejiang Province

Wenzhou Basic Medical and Health Technology Project

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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