Discovery of an Orally Efficacious MYC Inhibitor for Liver Cancer Using a GNMT-Based High-Throughput Screening System and Structure–Activity Relationship Analysis

Author:

Kant Rajni1ORCID,Yang Ming-Hui2,Tseng Chih-Hua34,Yen Chia-Hung56ORCID,Li Wei-You1,Tyan Yu-Chang7,Chen Marcelo8,Tzeng Cherng-Chyi9,Chen Wei-Cheng1,You Kaiting1,Wang Wen-Chieh10,Chen Yeh-Long49,Chen Yi-Ming Arthur1

Affiliation:

1. Graduate Institute of Biomedical and Pharmaceutical Science, Fu Jen Catholic University, New Taipei City 24205, Taiwan

2. Department of Medical Education and Research, Kaohsiung Veterans General Hospital, Kaohsiung 81362, Taiwan

3. School of Pharmacy, College of Pharmacy, Kaohsiung Medical University, Kaohsiung 807, Taiwan

4. Drug Development and Value Creation Research Center, Kaohsiung Medical University, Kaohsiung 80708, Taiwan

5. Graduate Institute of Natural Products, College of Pharmacy, Kaohsiung Medical University, Kaohsiung 80708, Taiwan

6. Research Center for Natural Products and Drug Development, Kaohsiung Medical University, Kaohsiung 80708, Taiwan

7. Department of Medical Imaging and Radiological Sciences, Kaohsiung Medical University, Kaohsiung 80708, Taiwan

8. Department of Urology, Mackay Memorial Hospital, Taipei 10449, Taiwan

9. Department of Medicinal and Applied Chemistry, College of Life Science, Kaohsiung Medical University, Kaohsiung 80708, Taiwan

10. Institute of Biotechnology and Pharmaceutical Research, National Health Research Institutes, 35 Keyan Road, Zhunan, Miaoli County 35053, Taiwan

Funder

Ministry of Health and Welfare

Ministry of Education

National Health Research Institutes

Universit??t zu K??ln

Kaohsiung Veterans General Hospital

Academia Sinica

Kaohsiung Medical University

Ministry of Science and Technology, Taiwan

KMU Global Networking Talent Plan

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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