Hypothesis-Driven, Structure-Based Design in Photopharmacology: The Case of eDHFR Inhibitors

Author:

Kobauri Piermichele1,Galenkamp Nicole S.2,Schulte Albert M.1ORCID,de Vries Jisk1,Simeth Nadja A.13ORCID,Maglia Giovanni2ORCID,Thallmair Sebastian45,Kolarski Dušan16,Szymanski Wiktor17ORCID,Feringa Ben L.1ORCID

Affiliation:

1. Stratingh Institute for Chemistry, University of Groningen, Nijenborgh 4, 9747 AG Groningen, The Netherlands

2. Groningen Biomolecular Science and Biotechnology Institute, University of Groningen, Nijenborgh 4, 9747 AG Groningen, The Netherlands

3. Institute for Organic and Biomolecular Chemistry, University of Goettingen, Tammannstr. 2, 37077 Göttingen, Germany

4. Groningen Biomolecular Sciences and Biotechnology Institute and Zernike Institute for Advanced Materials, University of Groningen, Nijenborgh 7, 9747 AG Groningen, The Netherlands

5. Frankfurt Institute for Advanced Studies, Ruth-Moufang-Straße 1, 60438 Frankfurt am Main, Germany

6. DWI-Leibniz Institut für interaktive Materialien e.V., RWTH Aachen University, Forckenbeckstraße 50, 52074 Aachen, Germany

7. Department of Radiology, Medical Imaging Center, University of Groningen, University Medical Center Groningen, Hanzeplein 1, 9713 GZ Groningen, The Netherlands

Funder

H2020 Marie Sklodowska-Curie Actions

Alexander von Humboldt-Stiftung

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Center for Information Technology, University of Groningen

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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