Discovery of High-Affinity Inhibitors of the BPTF Bromodomain

Author:

Lu Tian123,Lu Haibo45,Duan Zhe56,Wang Jun5,Han Jie5,Xiao Senhao5,Chen HuanHuan7,Jiang Hao5,Chen Yu5,Yang Feng5,Li Qi5,Chen Dongying7,Lin Jin1,Li Bo5ORCID,Jiang Hualiang5,Chen Kaixian35,Lu Wenchao8ORCID,Lin Hua59ORCID,Luo Cheng1345ORCID

Affiliation:

1. School of Pharmacy, Fujian Medical University, Fuzhou 350122, China

2. Guizhou University of Traditional Chinese Medicine, Guiyang, Guizhou 550025, China

3. School of Chinese Materia Medica, Nanjing University of Chinese Medicine, 138 Xianlin Road, Nanjing 210023, China

4. School of Pharmacy, Fudan University, 826 Zhangheng Road, Shanghai 201203, China

5. The Chemical Biology Center, Drug Design and Discovery Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China

6. School of Pharmacy, Nanchang University, Nanchang 330006, China

7. Laboratory of Pharmaceutical Analysis, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Zhangjiang Hi-Tech Park, Shanghai, 201203, China

8. Stanford Cancer Institute, Stanford School of Medicine, Stanford University, Stanford, California 94305, United States

9. Biomedical Research Center of South China, College of Life Sciences, Fujian Normal University, Fuzhou 350117, China

Funder

Science and Technology Commission of Shanghai Municipality

National Natural Science Foundation of China

State Key Laboratory of Drug Research

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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