Discovery of Potent and Selective CDK9 Degraders for Targeting Transcription Regulation in Triple-Negative Breast Cancer

Author:

Wei Dan12,Wang Hanlin342ORCID,Zeng Qinghe12,Wang Wenjing12,Hao Bingbing4,Feng Xule1,Wang Peipei4,Song Ning42,Kan Weijuan4,Huang Guifang5,Zhou Xiaoyu1,Tan Minjia4ORCID,Zhou Yubo426,Huang Ruimin125ORCID,Li Jia34267,Chen Xiao-Hua127ORCID

Affiliation:

1. Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China

2. University of Chinese Academy of Sciences, Beijing 100049, China

3. College of Pharmacy, Fudan University, Shanghai 201203, China

4. State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China

5. School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing 210023, China

6. Zhongshan Institute for Drug Discovery, The Institutes of Drug Discovery and Development, CAS, Zhongshan, Guangdong 528400, China

7. School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou 310024, China

Funder

National Natural Science Foundation of China

The Science and Technology Commission of Shanghai Municipality, China

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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