A Comprehensive <i>In Vitro</i> Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors-Reference-Cited by-同舟云学术

A Comprehensive In Vitro Characterization of a New Class of Indole-Based Compounds Developed as Selective Haspin Inhibitors

Published:2024-07-22 Issue:15 Volume:67 Page:12711-12734
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Vestuto Vincenzo¹,Ciaglia Tania¹,Musella Simona¹,Di Sarno Veronica¹,Smaldone Gerardina¹,Di Matteo Francesca¹,Scala Maria Carmina¹,Napolitano Valeria¹,Miranda Maria Rosaria¹,Amodio Giuseppina²,Novi Sara¹,Pepe Giacomo¹^ORCID,Basilicata Manuela Giovanna³,Gazzillo Erica¹,Pace Simona¹,Gomez-Monterrey Isabel M.⁴^ORCID,Sala Marina¹^ORCID,Bifulco Giuseppe¹^ORCID,Tecce Mario Felice¹,Campiglia Pietro¹^ORCID,Ostacolo Carmine¹^ORCID,Lauro Gianluigi¹^ORCID,Manfra Michele⁵,Bertamino Alessia¹^ORCID

Affiliation:

1. Department of Pharmacy, University of Salerno, Via G. Paolo II 132 , Salerno , Fisciano 84084, Italy

2. Department of Medicine, Surgery and Dentistry “Scuola Medica Salernitana″, University of Salerno, Salerno , Baronissi 84034, Italy

3. Department of Advanced Medical and Surgical Science, University of Campania “Luigi Vanvitelli”, P.zza L. Miraglia 2, Naples 80138, Italy

4. Department of Pharmacy, University Federico II of Naples, Via D. Montesano 49 , Naples 80131, Italy

5. Department of Science, University of Basilicata, Via dell’Ateneo Lucano 10 , Potenza 85100, Italy

Funder

Ministero dell'Universit? e della Ricerca

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.4c00718

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