Structure-Based Design and Synthesis of Covalent Inhibitors for Deubiquitinase and Acetyltransferase ChlaDUB1 of <i>Chlamydia trachomatis</i>-Reference-Cited by-同舟云学术

Structure-Based Design and Synthesis of Covalent Inhibitors for Deubiquitinase and Acetyltransferase ChlaDUB1 of Chlamydia trachomatis

Published:2024-06-19 Issue:13 Volume:67 Page:10710-10742
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Zimmermann Thomas¹,Feng Jiachen²,de Campos Luana Janaína²,Knight Lindsey A.³,Schlötzer Jan⁴,Ramirez Yesid A.¹^ORCID,Schwickert Kevin⁵^ORCID,Zehe Markus¹^ORCID,Adler Thomas B.¹^ORCID,Schirmeister Tanja⁵,Kisker Caroline⁴^ORCID,Sotriffer Christoph¹,Conda-Sheridan Martin²^ORCID,Decker Michael¹^ORCID

Affiliation:

1. Pharmazeutische und Medizinische Chemie, Institut für Pharmazie und Lebensmittelchemie, Julius-Maximilians-Universität Würzburg (JMU), Am Hubland, 97074 Würzburg, Germany

2. Department of Pharmaceutical Sciences, College of Pharmacy, University of Nebraska Medical Center, Omaha, Nebraska 68198, United States

3. Department of Pathology, Microbiology and Immunology, University of Nebraska Medical Center, Omaha, Nebraska 68198, United States

4. Rudolf Virchow Center for Integrative and Translational Bioimaging, Institute for Structural Biology, Julius-Maximilians-Universität Würzburg (JMU), 97080 Wurzburg, Germany

5. Institute of Pharmaceutical and Biomedical Sciences (IPBS), Johannes Gutenberg University Mainz, Staudingerweg 5, 55128 Mainz, Germany

Funder

Deutsche Forschungsgemeinschaft

National Institute of General Medical Sciences

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.4c00230

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3. Chlamydia, gonorrhoea, trichomoniasis and syphilis: global prevalence and incidence estimates, 2016

4. Sexually Transmitted Infections

5. WHO. WHO Guidelines for the Treatment of Chlamydia trachomatis; WHO guidelines for the treatment of Chlamydia trachomatis, 2016. https://apps.who.int/iris/bitstream/handle/10665/246165/9789241549714-eng.pdf.

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1. Correlating Predicted Reactivities with Experimental Inhibition Data of Covalent ChlaDUB1 Inhibitors;ACS Medicinal Chemistry Letters;2024-09-10