Targeting NOX2 with Bivalent Small-Molecule p47phox–p22phox Inhibitors

Author:

Zang Jie1,Peters Felix1,Cambet Yves2,Cifuentes-Pagano Eugenia34,Hissabu Munira Mohamed Shishay1,Dustin Christopher M.34,Svensson Lars Henrik1,Olesen Martin Mariboe1,Poulsen Mathias Feldt Lomholt1,Jacobsen Stig1,Tuelung Pernille Sønderby1ORCID,Narayanan Dilip1,Langkilde Annette Eva1ORCID,Gajhede Michael1ORCID,Pagano Patrick J.34,Jaquet Vincent25,Vilhardt Frederik6,Bach Anders1ORCID

Affiliation:

1. Department of Drug Design and Pharmacology, Faculty of Health and Medical Sciences, University of Copenhagen, Universitetsparken 2, DK-2100 Copenhagen, Denmark

2. READS unit, Centre Médical Universitaire, University of Geneva, Geneva CH-1211, Switzerland

3. Pittsburgh Heart, Lung, Blood and Vascular Medicine Institute, University of Pittsburgh, Pittsburgh, Pennsylvania 15261, United States

4. Department of Pharmacology and ChemicalBiology, University of Pittsburgh, Pittsburgh, Pennsylvania 15261, United States

5. Department of Pathology and Immunology, Centre Médical Universitaire, University of Geneva, Geneva CH-1211, Switzerland

6. Institute of Cellular and Molecular Medicine, Faculty of Health and Medical Sciences, University of Copenhagen, Blegdamsvej 3, DK-2200 Copenhagen, Denmark

Funder

Novo Nordisk Fonden

China Scholarship Council

Gigtforeningen

Lundbeck Foundation

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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