Kinetics, Thermodynamics, and Structural Effects of Quinoline-2-Carboxylates, Zinc-Binding Inhibitors of New Delhi Metallo-β-lactamase-1 Re-sensitizing Multidrug-Resistant Bacteria for Carbapenems

Author:

Jia Yuwen1,Schroeder Barbara1,Pfeifer Yvonne2,Fröhlich Christopher3,Deng Lihua1,Arkona Christoph1,Kuropka Benno4,Sticht Jana4,Ataka Kenichi5,Bergemann Silke1,Wolber Gerhard1ORCID,Nitsche Christoph6ORCID,Mielke Martin7,Leiros Hanna-Kirsti S.3,Werner Guido2,Rademann Jörg1ORCID

Affiliation:

1. Institute of Pharmacy, Freie Universität Berlin, Königin-Luise-Str. 2+4, Berlin 14195, Germany

2. FG13 Nosocomial Pathogens and Antibiotic Resistances, Department of Infectious Diseases, Robert Koch Institute, Burgstraße 37, Wernigerode 38855, Germany

3. Department of Chemistry, Faculty of Science and Technology, UiT The Arctic University of Norway, Tromsø 9037, Norway

4. Core Facility BioSupraMol, Institute for Chemistry and Biochemistry, Freie Universität Berlin, Thielallee 63, Berlin 14195, Germany

5. Department of Physics, Freie Universität Berlin, Arnimallee 14, Berlin 14195, Germany

6. Research School of Chemistry, Australian National University, Canberra 2601, Australian Capital Territory, Australia

7. Department of Infectious Diseases, Robert Koch Institute, Nordufer 20, Berlin 13353, Germany

Funder

Deutsche Forschungsgemeinschaft

Universitetet i Tromsø

China Scholarship Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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