Structure-Guided Design of a Domain-Selective Bromodomain and Extra Terminal N-Terminal Bromodomain Chemical Probe
Author:
Affiliation:
1. GSK, Medicines Research Centre, Stevenage SG1 2NY, Hertfordshire, U.K.
2. Department of Pure and Applied Chemistry, University of Strathclyde, Thomas Graham Building, 295 Cathedral Street, Glasgow G1 1XL, U.K.
Funder
Engineering and Physical Sciences Research Council
GlaxoSmithKline
University of Strathclyde
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.jmedchem.3c00906
Reference56 articles.
1. Histone Recognition and Large-Scale Structural Analysis of the Human Bromodomain Family
2. Bromodomain biology and drug discovery
3. BET domain co-regulators in obesity, inflammation and cancer
4. Bromodomain Histone Readers and Cancer
5. Bromodomain inhibition of the transcriptional coactivators CBP/EP300 as a therapeutic strategy to target the IRF4 network in multiple myeloma
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