N-(2-Aminophenyl)-benzamide Inhibitors of Class I HDAC Enzymes with Antiproliferative and Antifibrotic Activity

Author:

Gerokonstantis Dimitrios Triantafyllos12,Mantzourani Christiana12,Gkikas Dimitrios3,Wu Kai-Chen4,Hoang Huy N.4,Triandafillidi Ierasia12,Barbayianni Ilianna5,Kanellopoulou Paraskevi5,Kokotos Alexandros C.3,Moutevelis-Minakakis Panagiota12,Aidinis Vassilis5ORCID,Politis Panagiotis K.36,Fairlie David P.4ORCID,Kokotos George12

Affiliation:

1. Department of Chemistry, National and Kapodistrian University of Athens, Panepistimiopolis, Athens 15771, Greece

2. Center of Excellence for Drug Design and Discovery, National and Kapodistrian University of Athens, Panepistimiopolis, Athens 15771, Greece

3. Center of Basic Research, Biomedical Research Foundation of the Academy of Athens, Athens 11527, Greece

4. Institute for Molecular Bioscience, University of Queensland, Brisbane, Queensland 4072, Australia

5. Institute for Fundamental Biomedical Research, Biomedical Sciences Research Center “Alexander Fleming”, Athens 16672, Greece

6. School of Medicine, European University Cyprus, Nicosia 1516, Cyprus

Funder

European Commission

National Health and Medical Research Council

Australian Research Council

Hellenic Foundation for Research and Innovation

Stavros Niarchos Foundation

Government of Greece

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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