Design and Syntheses of Highly Potent Teixobactin Analogues against Staphylococcus aureus, Methicillin-Resistant Staphylococcus aureus (MRSA), and Vancomycin-Resistant Enterococci (VRE) in Vitro and in Vivo

Author:

Parmar Anish,Lakshminarayanan Rajamani1,Iyer Abhishek2,Mayandi Venkatesh1,Leng Goh Eunice Tze1,Lloyd Daniel G.,Chalasani Madhavi Latha S.3,Verma Navin K.13,Prior Stephen H.,Beuerman Roger W.1,Madder Annemieke2ORCID,Taylor Edward J.,Singh IshwarORCID

Affiliation:

1. Singapore Eye Research Institute, The Academia, Discovery Tower Level 6, 20 College Road, 169857 Singapore

2. Organic and Biomimetic Chemistry Research Group, Department of Organic and Macromolecular Chemistry, Ghent University, Krijgslaan 281 (S4), Ghent B-9000, Belgium

3. Lee Kong Chian School of Medicine, Nanyang Technological University, 636921 Singapore

Funder

Royal Society

Ministry of Education - Singapore

National Medical Research Council

Lincoln University

H2020 Marie Sklodowska-Curie Actions

Rosetrees Trust

Lee Kong Chian School of Medicine, Nanyang Technological University

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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