Allosteric Inhibitors of SHP2 with Therapeutic Potential for Cancer Treatment

Author:

Xie Jingjing12,Si Xiaojia3,Gu Shoulai1,Wang Mingliang4,Shen Jian12,Li Haoyan12,Shen Jian5,Li Dan6,Fang Yanjia1,Liu Cong1,Zhu Jidong1

Affiliation:

1. Interdisciplinary Research Center on Biology and Chemistry, Center for Excellence in Molecular Synthesis, Shanghai Institute of Organic Chemistry, Chinese Academy of Sciences, 26 Qiuyue Road, Shanghai 201203, China

2. University of the Chinese Academy of Sciences, 19 A Yuquan Road, Shijingshan District, Beijing 100049, China

3. Organisch-Chemisches Institut, Ruprecht-Karls-Universität Heidelberg, Im Neuenheimer Feld 270, 69120 Heidelberg, Germany

4. Department of Natural Products Chemistry, Fudan University, 826 Zhangheng Road, Shanghai 201203, China

5. Viva Biotech Ltd. 334 Aidisheng Road, Shanghai 201203, China

6. Key Laboratory for the Genetics of Developmental and Neuropsychiatric Disorders (Ministry of Education), Bio-X Institutes, Shanghai Jiao Tong University, Shanghai 200240, China

Funder

Ministry of Science and Technology of the People's Republic of China

Science and Technology Commission of Shanghai Municipality

Chinese Academy of Sciences

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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