1. Mount Sinai Center for Therapeutics Discovery, Departments of Pharmacological Sciences and Oncological Sciences, Tisch Cancer Institute, Icahn School of Medicine at Mount Sinai, New York, New York 10029, United States
2. Structural Genomics Consortium, University of Toronto, Toronto, Ontario M5G 1L7, Canada
3. Ontario Institute for Cancer Research, Toronto, Ontario M5G 0A3, Canada
4. Eli Lilly and Company, Lilly Research Laboratories, Indianapolis, Indiana 46225, United States
5. Department of Medical Biophysics, University of Toronto, Toronto, Ontario M5G 1L7, Canada
6. Department of Pharmacology and Toxicology, University of Toronto, Toronto, Ontario M5S 1A8, Canada