1,4-Dihydropyridines Active on the SIRT1/AMPK Pathway Ameliorate Skin Repair and Mitochondrial Function and Exhibit Inhibition of Proliferation in Cancer Cells

Author:

Valente Sergio1,Mellini Paolo1,Spallotta Francesco2,Carafa Vincenzo3,Nebbioso Angela3,Polletta Lucia4,Carnevale Ilaria4,Saladini Serena4,Trisciuoglio Daniela5,Gabellini Chiara5,Tardugno Maria1,Zwergel Clemens1,Cencioni Chiara2,Atlante Sandra2,Moniot Sébastien6,Steegborn Clemens6,Budriesi Roberta7,Tafani Marco4,Del Bufalo Donatella5,Altucci Lucia38,Gaetano Carlo2,Mai Antonello19

Affiliation:

1. Department of Drug Chemistry and Technologies, Sapienza University of Rome, P. le A. Moro 5, 00185 Rome, Italy

2. Division of Cardiovascular Epigenetics, Department of Cardiology, Goethe University, Theodor-Stern-Kai 7, 60590 Frankfurt am Main, Germany

3. Department of Biochemistry, Biophysics and General Pathology, Second University of Naples, Vico L. De Crecchio 7, 80138 Naples, Italy

4. Department of Experimental Medicine, Sapienza University of Rome, Viale Regina Elena 324, 00161 Rome, Italy

5. Regina Elena National Cancer Institute, Via Elio Chianesi, 53, 00144 Rome, Italy

6. Department of Biochemistry, University of Bayreuth; 95447 Bayreuth, Germany

7. Department of Pharmacy and Biotechnology, University of Bologna, Via Zamboni 33, 40126 Bologna, Italy

8. Institute of Genetics and Biophysics, IGB, Adriano Buzzati Traverso, Via P. Castellino 111, 80131 Naples, Italy

9. Pasteur Institute, Cenci-Bolognetti Foundation, Sapienza University of Rome, P. le A. Moro 5, 00185 Rome, Italy

Funder

Associazione Italiana per la Ricerca sul Cancro

Fondazione Umberto Veronesi

Seventh Framework Programme

Ministero dell'Istruzione, dell'Università e della Ricerca

Istituto Italiano di Tecnologia

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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