First-in-Class Dual Hybrid Carbonic Anhydrase Inhibitors and Transient Receptor Potential Vanilloid 1 Agonists Revert Oxaliplatin-Induced Neuropathy

Author:

Angeli Andrea1ORCID,Micheli Laura2,Carta Fabrizio1ORCID,Ferraroni Marta3ORCID,Pirali Tracey4ORCID,Fernandez Carvajal Asia5,Ferrer Montiel Antonio5,Di Cesare Mannelli Lorenzo2,Ghelardini Carla2,Supuran Claudiu T.1ORCID

Affiliation:

1. NEUROFARBA Department, Sezione di Scienze Farmaceutiche, University of Florence, via Ugo Schiff 6, 50019 Sesto Fiorentino, Florence, Italy

2. Pharmacology and Toxicology Section, Department of Neuroscience, Psychology, Drug Research and Child Health (NEUROFARBA), University of Florence, viale Gaetano Pieraccini 6, 50139 Firenze, Florence, Italy

3. Department of Chemistry ″Ugo Schiff″, University of Florence, via della Lastruccia 3-13, I-50019 Sesto Fiorentino, Italy

4. Dipartimento Di Scienze del Farmaco, Università Degli Studi del Piemonte Orientale, 28100 Novara, Italy

5. Instituto de Investigación, Desarrollo e Innovación en Biotecnología Sanitaria de Elche (IDiBE), Universitas Miguel Hernández, 03202 Elche, Spain

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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