Design and Synthesis of Triazole-Containing HDAC Inhibitors That Induce Antitumor Effects and Immune Response

Author:

Sun Nan12,Yang Kexin34,Yan Wenzhong2,Yao Mingyue345,Yu Chengcheng6,Duan Wenwen2,Gu Xiaoke1,Guo Dong1ORCID,Jiang Hualiang347,Xie Chengying347,Cheng Jianjun24ORCID

Affiliation:

1. Jiangsu Key Laboratory of New Drug Research and Clinical Pharmacy, Xuzhou Medical University, Xuzhou 221004, Jiangsu, China

2. iHuman Institute, ShanghaiTech University, Shanghai 201210, China

3. Shanghai Institute for Advanced Immunochemical Studies, ShanghaiTech University, Shanghai 201210, China

4. School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China

5. The First Affiliated Hospital of USTC (Anhui Provincial Hospital), Division of Life Sciences and Medicine, University of Science and Technology of China, Hefei 230001, Anhui, China

6. Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China

7. Lingang Laboratory, Shanghai 200031, China

Funder

Shanghai Municipal People's Government

ShanghaiTech University

Lingang Laboratory

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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