Chemo- and Site-Selective Lysine Modification of Peptides and Proteins under Native Conditions Using the Water-Soluble Zolinium

Author:

Sun Haiguo12,Xi Mengyu12,Jin Qiang3,Zhu Zhengdan12ORCID,Zhang Yani3,Jia Guihua3,Zhu Guanghao3,Sun Mengru3,Zhang Hongwei3,Ren Xuelian12,Zhang Yong12,Xu Zhijian12ORCID,Huang He12ORCID,Shen Jingshan12ORCID,Li Bo124ORCID,Ge Guangbo3,Chen Kaixian132,Zhu Weiliang132ORCID

Affiliation:

1. CAS Key Laboratory of Receptor Research, State Key Laboratory of Drug Research; Drug Discovery and Design Center, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, 555 Zuchongzhi Road, Shanghai 201203, China

2. School of Pharmacy, University of Chinese Academy of Sciences, No. 19A Yuquan Road, Beijing 100049, China

3. Shanghai Frontiers Science Center of TCM Chemical Biology; Institute of Interdisciplinary Integrative Medicine Research, Shanghai University of Traditional Chinese Medicine, 1200 Cailun Road, Shanghai 201203, China

4. State Key Laboratory of Natural and Biomimetic Drugs, Peking University, No. 38 Xue Yuan Road, Haidian District, Beijing 100191, China

Funder

Natural Science Foundation of Shanghai

Ministry of Science and Technology of the People's Republic of China

National Natural Science Foundation of China

Shanghai Talent Development Fund

State Key Laboratory of Natural and Biomimetic Drugs, Peking University

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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