Discovery of Benzoylsulfonohydrazides as Potent Inhibitors of the Histone Acetyltransferase KAT6A

Author:

Leaver David J.,Cleary Benjamin,Nguyen Nghi,Priebbenow Daniel L.ORCID,Lagiakos H. Rachel1,Sanchez Julie23,Xue Lian4,Huang Fei4,Sun Yuxin,Mujumdar Prashant,Mudududdla Ramesh,Varghese Swapna,Teguh Silvia,Charman Susan A.,White Karen L.,Katneni Kasiram,Cuellar Matthew5,Strasser Jessica M.5,Dahlin Jayme L.6,Walters Michael A.5ORCID,Street Ian P.213,Monahan Brendon J.213,Jarman Kate E.23,Sabroux Helene Jousset23,Falk Hendrik213,Chung Matthew C.7,Hermans Stefan J.7,Parker Michael W.7,Thomas Tim23,Baell Jonathan B.48ORCID

Affiliation:

1. Cancer Therapeutics CRC, 343 Royal Parade, Parkville, Victoria 3052, Australia

2. Walter and Eliza Hall Institute of Medical Research, 1G Royal Parade, Parkville, Victoria 3052, Australia

3. Department of Medical Biology, University of Melbourne, Parkville, Victoria 3050, Australia

4. School of Pharmaceutical Sciences, Nanjing Tech University, No. 30 South Puzhu Road, Nanjing 211816, People’s Republic of China

5. Institute for Therapeutics Discovery and Development, University of Minnesota, 717 Delaware Street SE, Minneapolis, Minnesota 55455, United States

6. Department of Pathology, Brigham and Women’s Hospital, Boston, 75 Francis Street, Boston, Massachusetts 02115, United States

7. ACRF Rational Drug Discovery Centre, St. Vincent’s Institute of Medical Research, Fitzroy, Victoria 3065, Australia

8. ARC Centre for Fragment-Based Design, Monash University, Parkville, Victoria 3052, Australia

Funder

National Health and Medical Research Council

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

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