Novel Alaninamide Derivatives with Drug-like Potential for Development as Antiseizure and Antinociceptive Therapies─In Vitro and In Vivo Characterization

Author:

Jakubiec Marcin1,Abram Michał1ORCID,Zagaja Mirosław2,Andres-Mach Marta2,Szala-Rycaj Joanna2,Latacz Gniewomir3,Honkisz-Orzechowska Ewelina3,Mogilski Szczepan4,Kubacka Monika4,Szafarz Małgorzata5,Pociecha Krzysztof5,Przejczowska-Pomierny Katarzyna5,Wyska Elżbieta5ORCID,Socała Katarzyna6,Nieoczym Dorota6,Szulczyk Bartłomiej7,Wlaź Piotr6ORCID,Metcalf Cameron S.8ORCID,Wilcox Karen8,Kamiński Rafał M.1,Kamiński Krzysztof1ORCID

Affiliation:

1. Department of Medicinal Chemistry, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland

2. Department of Experimental Pharmacology, Institute of Rural Health, Jaczewskiego 2, 20-950 Lublin, Poland

3. Department of Technology and Biotechnology of Drugs, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland

4. Department Pharmacodynamics, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland

5. Department of Pharmacokinetics and Physical Pharmacy, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Krakow, Poland

6. Department of Animal Physiology and Pharmacology, Institute of Biological Sciences, Faculty of Biology and Biotechnology, Maria Curie-Skłodowska University, Akademicka 19, 20-033 Lublin, Poland

7. Chair and Department of Pharmacotherapy and Pharmaceutical Care, Centre for Preclinical Research and Technology, Medical University of Warsaw, Banacha 1B, 02-097 Warsaw, Poland

8. Department of Pharmacology and Toxicology, University of Utah, Salt Lake City, Utah 84112, United States

Funder

Narodowe Centrum Nauki

Publisher

American Chemical Society (ACS)

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