Molecular-Interaction and Signaling Profiles of AM3677, a Novel Covalent Agonist Selective for the Cannabinoid 1 Receptor-Reference-Cited by-同舟云学术

Molecular-Interaction and Signaling Profiles of AM3677, a Novel Covalent Agonist Selective for the Cannabinoid 1 Receptor

Published:2015-05-29 Issue:8 Volume:6 Page:1400-1410
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Janero David R.¹,Yaddanapudi Suma¹,Zvonok Nikolai¹,Subramanian Kumar V.¹,Shukla Vidyanand G.¹,Stahl Edward²,Zhou Lei²,Hurst Dow³,Wager-Miller James⁴,Bohn Laura M.²,Reggio Patricia H.³,Mackie Ken⁴,Makriyannis Alexandros¹

Affiliation:

1. Center for Drug Discovery and Departments of Chemistry and Chemical Biology and Pharmaceutical Sciences, Northeastern University, Boston, Massachusetts 02115, United States

2. Departments of Molecular Therapeutics and Neuroscience, Scripps Research Institute, Jupiter, Florida 33458, United States

3. Center for Drug Discovery, University of North Carolina at Greensboro, Greensboro, North Carolina 27402, United States

4. Department of Psychological and Brain Sciences, Indiana University, Bloomington, Indiana 47405, United States

Funder

National Institute on Drug Abuse

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/acschemneuro.5b00090

Reference65 articles.

1. The endocannabinoid system: Its general strategy of action, tools for its pharmacological manipulation and potential therapeutic exploitation

2. Cannabinoid receptors: nomenclature and pharmacological principles

3. The Endocannabinoid System and the Brain

4. Endocannabinoid-mediated retrograde modulation of synaptic transmission

5. Endocannabinoid system dysfunction in mood and related disorders

Cited by 22 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Recent advances in the development of CB1R selective probes;Frontiers in Natural Products;2023-07-18

2. Large library docking for cannabinoid-1 receptor agonists with reduced side effects;2023-03-03

3. Differential Enantiomer-Specific Signaling of Cannabidiol at CB₁Receptors;Molecular Pharmacology;2022-09-24

4. Oxa-adamantyl cannabinoids;Bioorganic & Medicinal Chemistry Letters;2021-04

5. Novel Functionalized Cannabinoid Receptor Probes: Development of Exceptionally Potent Agonists;Journal of Medicinal Chemistry;2021-03-24