6,7-Dihydro-2-benzothiophen-4(5H)-ones: A Novel Class of GABA-A α5 Receptor Inverse Agonists-Reference-Cited by-同舟云学术

6,7-Dihydro-2-benzothiophen-4(5H)-ones: A Novel Class of GABA-A α5 Receptor Inverse Agonists

Published:2002-02-12 Issue:6 Volume:45 Page:1176-1179
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Chambers Mark S.¹,Atack John R.¹,Bromidge Frances A.¹,Broughton Howard B.¹,Cook Susan¹,Dawson Gerard R.¹,Hobbs Sarah C.¹,Maubach Karen A.¹,Reeve Austin J.¹,Seabrook Guy R.¹,Wafford Keith¹,MacLeod Angus M.¹

Affiliation:

1. Merck Sharp & Dohme Research Laboratories, The Neuroscience Research Centre, Terlings Park, Eastwick Road, Harlow, Essex CM20 2QR, U.K.

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm010471b

Reference39 articles.

1. Olsen, R. W.; Venter J. C.Benzodiazepine/GABA receptors and chloridechannels: Structural and functional properties; Alan R. Liss Inc. New York, 1986.

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