1. Chemistry Research Laboratory, University of Oxford, 12 Mansfield Road, Oxford OX1 3TA, United Kingdom
2. Pfizer Worldwide Research and Development, Groton, Connecticut 06340, United States
3. Discovery Chemistry, Janssen Research and Development, Jarama 75A, Toledo E-45007, Spain
4. Univ. Lyon, Université Lyon I, CNRS, INSA, CPE-Lyon, ICBMS, UMR 5246, 1 Rue Victor Grignard, 69622 Villeurbanne cedex, France
5. Micro Flow Chemistry and Synthetic Methodology, Department of Chemical Engineering and Chemistry, Eindhoven University of Technology, Het Kranenveld, Bldg 14, Helix, 5600 MB Eindhoven, The Netherlands
6. Global Chemistry, UCB New Medicines, UCB Biopharma Sprl, 1420 Braine-L’Alleud, Belgium