Dissimilar Effect of P-Glycoprotein and Breast Cancer Resistance Protein Inhibition on the Distribution of Erlotinib to the Retina and Brain in Humans and Mice

Author:

Biali Myriam El1,Auvity Sylvain23,Cisternino Salvatore23,Smirnova Maria2,Hacker Marcus4,Zeitlinger Markus1,Mairinger Severin14,Tournier Nicolas5,Bauer Martin1,Langer Oliver14ORCID

Affiliation:

1. Department of Clinical Pharmacology, Medical University of Vienna, 1090 Vienna, Austria

2. Inserm UMRS1144, Optimisation Thérapeutique en Neuropsychopharmacologie, Université Paris Cité, F-75006 Paris, France

3. Service Pharmacie, Assistance Publique-Hôpitaux de Paris, Hôpital Universitaire-Necker-Enfants Malades, F-75015 Paris, France

4. Division of Nuclear Medicine, Department of Biomedical Imaging and Image-guided Therapy, Medical University of Vienna, 1090 Vienna, Austria

5. Laboratoire d’Imagerie Biomédicale Multimodale (BioMaps), CEA, CNRS, Inserm, Service Hospitalier Frédéric Joliot, Université Paris-Saclay, 91401 Orsay, France

Funder

Austrian Science Fund

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Pharmaceutical Science,Molecular Medicine

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