Fluorescence Linked Enzyme Chemoproteomic Strategy for Discovery of a Potent and Selective DAPK1 and ZIPK Inhibitor-Reference-Cited by-同舟云学术

Fluorescence Linked Enzyme Chemoproteomic Strategy for Discovery of a Potent and Selective DAPK1 and ZIPK Inhibitor

Published:2013-10-17 Issue:12 Volume:8 Page:2715-2723
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Carlson David A.¹,Franke Aaron S.²,Weitzel Douglas H.¹,Speer Brittany L.¹,Hughes Philip F.¹,Hagerty Laura¹,Fortner Christopher N.¹,Veal James M.³,Barta Thomas E.¹,Zieba Bartosz J.²,Somlyo Avril V.²,Sutherland Cindy⁴,Deng Jing Ti⁴,Walsh Michael P.⁴,MacDonald Justin A.⁴,Haystead Timothy A. J.¹

Affiliation:

1. Department of Pharmacology and Cancer Biology, Duke University Medical Center, Durham, North Carolina 27710, United States

2. Department of Molecular Physiology and Biological Physics, University of Virginia, Charlottesville, Virginia 22908, United States

3. Quanticel Pharmaceuticals, San Francisco, California 94158, United States

4. Smooth Muscle Research Group at the Libin Cardiovascular Institute of Alberta. Department of Biochemistry & Molecular Biology, University of Calgary, 3280 Hospital Drive NW, Calgary, AB T2N 4Z6, Canada

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cb400407c

Reference47 articles.

1. The Death-Associated Protein Kinases: Structure, Function, and Beyond

2. DAPk Protein Family and Cancer

3. ZIP kinase, a key regulator of myosin protein phosphatase 1

4. Targeting protein kinases in central nervous system disorders

5. Deletion of the Kinase Domain in Death-Associated Protein Kinase Attenuates Tubular Cell Apoptosis in Renal Ischemia-Reperfusion Injury

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