Discovery of 5-[5-Fluoro-2-oxo-1,2- dihydroindol-(3Z)-ylidenemethyl]-2,4- dimethyl-1H-pyrrole-3-carboxylic Acid (2-Diethylaminoethyl)amide, a Novel Tyrosine Kinase Inhibitor Targeting Vascular Endothelial and Platelet-Derived Growth Factor Receptor Tyrosine Kinase
Author:
Affiliation:
1. SUGEN, Inc., 230 E. Grand Avenue, South San Francisco, California 94080
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm0204183
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2. VEGF: an update on biological and therapeutic aspects
3. Evidence for Distinct Signaling Properties and Biological Responses Induced by the PDGF Receptor α and β Subtypes
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