X-ray Structural and Biological Evaluation of a Series of Potent and Highly Selective Inhibitors of Human Coronavirus Papain-like Proteases-Reference-Cited by-同舟云学术

X-ray Structural and Biological Evaluation of a Series of Potent and Highly Selective Inhibitors of Human Coronavirus Papain-like Proteases

Published:2014-03-14 Issue:6 Volume:57 Page:2393-2412
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Báez-Santos Yahira M.¹,Barraza Scott J.²,Wilson Michael W.²,Agius Michael P.²,Mielech Anna M.³,Davis Nicole M.¹,Baker Susan C.³,Larsen Scott D.²,Mesecar Andrew D.¹

Affiliation:

1. Department of Biological Sciences, Purdue University, 915 W. State Street, West Lafayette, Indiana 47907, United States

2. Vahlteich Medicinal Chemistry Core and Department of Medicinal Chemistry, College of Pharmacy, University of Michigan, Ann Arbor, Michigan 48109, United States

3. Department of Microbiology and Immunology, Loyola University Chicago Stritch School of Medicine, Maywood, Illinois 60153, United States

Funder

National Institutes of Health

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm401712t

Reference43 articles.

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2. avan Boheemen, S.; Zaki, A. M.; Bestebroer,T. M.; de Graaf, M.; Victor, S.; Osterhaus, A. D.; Haagmans, B. L.; Fouchier, R. A.Genomic Analysis for a Newly Isolated Human Betacoronavirus Lineage 2C. Submitted Sep 26, 2012.

3. Severe respiratory illness caused by a novel coronavirus, in a patient transferred to the United Kingdom from the Middle East, September 2012

4. The United Kingdom public health response to an imported laboratory confirmed case of a novel coronavirus in September 2012

5. Middle East Respiratory Syndrome Coronavirus (MERS-CoV): Announcement of the Coronavirus Study Group

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