Stereospecific High-affinity TRPV1 Antagonists: Chiral N-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide Analogues-Reference-Cited by-同舟云学术

Stereospecific High-affinity TRPV1 Antagonists: Chiral N-(2-Benzyl-3-pivaloyloxypropyl) 2-[4-(methylsulfonylamino)phenyl]propionamide Analogues

Published:2007-12-12 Issue:1 Volume:51 Page:57-67
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Ryu HyungChul¹,Jin Mi-Kyoung¹,Kim Su Yeon¹,Choi Hyun-Kyung¹,Kang Sang-Uk¹,Kang Dong Wook¹,Lee Jeewoo¹,Pearce Larry V.¹,Pavlyukovets Vladimir A.¹,Morgan Matthew A.¹,Tran Richard¹,Toth Attila¹,Lundberg Daniel J.¹,Blumberg Peter M.¹

Affiliation:

1. Research Institute of Pharmaceutical Sciences, College of Pharmacy, Seoul National University, Shinlim-Dong, Kwanak-Ku, Seoul 151-742, Korea, and Laboratory of Cancer Biology and Genetics, Center for Cancer Research, National Cancer Institute, National Institutes of Health, Bethesda, Maryland 20892

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm701049p

Reference18 articles.

1. The diversity in the vanilloid (TRPV) receptor family of ion channels

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5. Impaired Nociception and Pain Sensation in Mice Lacking the Capsaicin Receptor

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