Protein Arginine Deiminase 2 Binds Calcium in an Ordered Fashion: Implications for Inhibitor Design

Author:

Slade Daniel J.12,Fang Pengfei3,Dreyton Christina J.14,Zhang Ying5,Fuhrmann Jakob1,Rempel Don5,Bax Benjamin D.6,Coonrod Scott A.7,Lewis Huw D.8,Guo Min3,Gross Michael L.5,Thompson Paul R.14

Affiliation:

1. Department of Chemistry, The Scripps Research Institute, Jupiter, Florida 33458, United States

2. Department of Biochemistry, Virginia Polytechnic Institute and State University, Blacksburg, Virginia 24061, United States

3. Department of Cancer Biology, The Scripps Research Institute, Jupiter, Florida 33458, United States

4. Department of Biochemistry and Molecular Pharmacology, University of Massachusetts Medical School, Worcester, Massachusetts 01605, United States

5. Department of Chemistry, Washington University in St. Louis, St. Louis, Missouri 63130, United States

6. Molecular Discovery Research, GlaxoSmithKline, Medicines Research Centre, Gunnels Wood Road, Stevenage, Herts., SG1 2NY, United Kingdom

7. Department of Biomedical Sciences, Baker Institute for Animal Health, Cornell University, Ithaca, New York 14853, United States

8. EpiNova DPU, Immuno-Inflammation Therapy Area, GlaxoSmithKline, Medicines Research Centre, Gunnels Wood Road, Stevenage, Herts., SG1 2NY, United Kingdom

Funder

U.S. Department of Defense

National Institute of General Medical Sciences

The Scripps Research Institute

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

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